Opioid analgesics


Opioid analgesics are a subcategory of pharmaceutical Active Pharmaceutical Ingredients (APIs) that are commonly used for pain management. These potent substances interact with specific receptors in the central nervous system, producing analgesic effects and reducing the perception of pain. Opioid analgesics are derived from opium alkaloids or synthetic compounds that mimic their effects. They are classified based on their strength, with some being classified as strong opioids (e.g., morphine, fentanyl) and others as weak opioids (e.g., codeine, tramadol). These APIs work by binding to opioid receptors, primarily located in the brain, spinal cord, and gastrointestinal tract. By activating these receptors, opioid analgesics modulate pain signals, resulting in pain relief. Additionally, they can induce feelings of euphoria, sedation, and respiratory depression, which can be both beneficial and potentially harmful.

Due to their potency and potential for abuse, opioid analgesics are tightly regulated substances. They are primarily prescribed for acute and chronic pain management, such as post-surgical pain, cancer pain, and severe injuries. However, their misuse and addiction potential have led to a public health crisis in many countries.

In conclusion, opioid analgesics are a subcategory of pharmaceutical APIs that play a crucial role in pain management. While they provide effective pain relief, their use requires careful monitoring and adherence to prescribing guidelines to mitigate the risks associated with their potential for abuse and addiction.

NameCAS numberCategoryAmount of suppliersAPI market price
14-hydroxycodeinone508-54-3Opioid analgesicsView 1 Suppliers Average price per kg: $
Alfentanil71195-58-9Opioid analgesicsView 6 Suppliers Average price per kg: $
Buprenorphine52485-79-7Opioid analgesicsView 32 Suppliers Average price per kg: $
Butorphanol42408-82-2Opioid analgesicsView 6 Suppliers Average price per kg: $
Codeine76-57-3Opioid analgesicsView 12 Suppliers Average price per kg: $
Codeine phosphate hemihydrateOpioid analgesicsView 22 Suppliers Average price per kg: $
Dezocine53648-55-8Opioid analgesicsView 1 Suppliers Average price per kg: $
Dihydrocodeine125-28-0Opioid analgesicsView 7 Suppliers Average price per kg: $
Ethylmorphine76-58-4Opioid analgesicsView 1 Suppliers Average price per kg: $
Etorphine14521-96-1Opioid analgesicsView 1 Suppliers Average price per kg: $
Fentanyl437-38-7Opioid analgesicsView 17 Suppliers Average price per kg: $
Hydrocodone125-29-1Opioid analgesicsView 11 Suppliers Average price per kg: $
Hydromorphone466-99-9Opioid analgesicsView 15 Suppliers Average price per kg: $
Levomethadone hydrochloride5967-73-7Opioid analgesicsView 6 Suppliers Average price per kg: $
Levorphanol77-07-6Opioid analgesicsView 2 Suppliers Average price per kg: $
Methadone76-99-3Opioid analgesicsView 21 Suppliers Average price per kg: $
Methyl nalbuphine90242-27-6Opioid analgesicsView 3 Suppliers Average price per kg: $
Morphine57-27-2Opioid analgesicsView 12 Suppliers Average price per kg: $
Morphine sulfateOpioid analgesicsView 10 Suppliers Average price per kg: $
N-Methylnorbuprenorphine 3-Methyl Ether16196-70-6Opioid analgesicsView 3 Suppliers Average price per kg: $
Nalbuphine20594-83-6Opioid analgesicsView 9 Suppliers Average price per kg: $
Nalbuphine hydrochloride23277-43-2Opioid analgesicsView 2 Suppliers Average price per kg: $
Noroxycodone57664-96-7Opioid analgesicsView 1 Suppliers Average price per kg: $
Noroxycodone hydrochloride52446-25-0Opioid analgesicsView 1 Suppliers Average price per kg: $
Noroxymorphone33522-95-1Opioid analgesicsView 4 Suppliers Average price per kg: $
Noroxymorphone hydrochloride52446-24-9Opioid analgesicsView 2 Suppliers Average price per kg: $
Opium tinctureOpioid analgesicsView 7 Suppliers Average price per kg: $
Oxycodone76-42-6Opioid analgesicsView 19 Suppliers Average price per kg: $
Oxymorphone76-41-5Opioid analgesicsView 5 Suppliers Average price per kg: $
Pentazocine359-83-1Opioid analgesicsView 4 Suppliers Average price per kg: $
Pethidine57-42-1Opioid analgesicsView 7 Suppliers Average price per kg: $
Piritramide302-41-0Opioid analgesicsView 3 Suppliers Average price per kg: $
Remifentanil132875-61-7Opioid analgesicsView 11 Suppliers Average price per kg: $
Remifentanil hydrochloride132539-07-2Opioid analgesicsView 0 Suppliers Average price per kg: $
Sufentanil56030-54-7Opioid analgesicsView 8 Suppliers Average price per kg: $
Tapentadol175591-23-8Opioid analgesicsView 16 Suppliers Average price per kg: $
Tapentadol HydrochlorideOpioid analgesicsView 3 Suppliers Average price per kg: $
Thebaine115-37-7Opioid analgesicsView 1 Suppliers Average price per kg: $
Tilidine hydrochloride hemihydrate255733-17-6Opioid analgesicsView 4 Suppliers Average price per kg: $
Tramadol27203-92-5Opioid analgesicsView 51 Suppliers Average price per kg: $