Opioid analgesics


Opioid analgesics are a subcategory of pharmaceutical Active Pharmaceutical Ingredients (APIs) that are commonly used for pain management. These potent substances interact with specific receptors in the central nervous system, producing analgesic effects and reducing the perception of pain. Opioid analgesics are derived from opium alkaloids or synthetic compounds that mimic their effects. They are classified based on their strength, with some being classified as strong opioids (e.g., morphine, fentanyl) and others as weak opioids (e.g., codeine, tramadol). These APIs work by binding to opioid receptors, primarily located in the brain, spinal cord, and gastrointestinal tract. By activating these receptors, opioid analgesics modulate pain signals, resulting in pain relief. Additionally, they can induce feelings of euphoria, sedation, and respiratory depression, which can be both beneficial and potentially harmful.

Due to their potency and potential for abuse, opioid analgesics are tightly regulated substances. They are primarily prescribed for acute and chronic pain management, such as post-surgical pain, cancer pain, and severe injuries. However, their misuse and addiction potential have led to a public health crisis in many countries.

In conclusion, opioid analgesics are a subcategory of pharmaceutical APIs that play a crucial role in pain management. While they provide effective pain relief, their use requires careful monitoring and adherence to prescribing guidelines to mitigate the risks associated with their potential for abuse and addiction.

NameCAS numberCategoryAmount of suppliers
14-hydroxycodeinone508-54-3Opioid analgesics1
Alfentanil71195-58-9Opioid analgesics6
Buprenorphine52485-79-7Opioid analgesics30
Butorphanol42408-82-2Opioid analgesics6
Codeine76-57-3Opioid analgesics12
Codeine phosphate hemihydrateOpioid analgesics22
Dezocine53648-55-8Opioid analgesics1
Dihydrocodeine125-28-0Opioid analgesics7
Ethylmorphine76-58-4Opioid analgesics1
Etorphine14521-96-1Opioid analgesics1
Fentanyl437-38-7Opioid analgesics17
Hydrocodone125-29-1Opioid analgesics11
Hydromorphone466-99-9Opioid analgesics15
Levomethadone hydrochloride5967-73-7Opioid analgesics5
Levorphanol77-07-6Opioid analgesics2
Methadone76-99-3Opioid analgesics21
Methyl nalbuphine90242-27-6Opioid analgesics3
Morphine57-27-2Opioid analgesics11
Morphine sulfateOpioid analgesics10
N-Methylnorbuprenorphine 3-Methyl Ether16196-70-6Opioid analgesics3
Nalbuphine20594-83-6Opioid analgesics9
Nalbuphine hydrochloride23277-43-2Opioid analgesics2
Noroxycodone57664-96-7Opioid analgesics1
Noroxycodone hydrochloride52446-25-0Opioid analgesics1
Noroxymorphone33522-95-1Opioid analgesics4
Noroxymorphone hydrochloride52446-24-9Opioid analgesics2
Opium tinctureOpioid analgesics6
Oxycodone76-42-6Opioid analgesics19
Oxymorphone76-41-5Opioid analgesics5
Pentazocine359-83-1Opioid analgesics4
Pethidine57-42-1Opioid analgesics7
Piritramide302-41-0Opioid analgesics3
Remifentanil132875-61-7Opioid analgesics11
Remifentanil hydrochloride132539-07-2Opioid analgesics0
Sufentanil56030-54-7Opioid analgesics8
Tapentadol175591-23-8Opioid analgesics16
Tapentadol HydrochlorideOpioid analgesics3
Thebaine115-37-7Opioid analgesics1
Tilidine hydrochloride hemihydrate255733-17-6Opioid analgesics4
Tramadol27203-92-5Opioid analgesics49