Protein kinase inhibitors


Protein kinase inhibitors are a vital subcategory of pharmaceutical active pharmaceutical ingredients (APIs) that play a crucial role in targeted cancer therapies. These inhibitors specifically target and block the activity of protein kinases, enzymes that regulate various cellular processes, including cell growth, division, and signal transduction.

Protein kinase inhibitors function by binding to the active site of protein kinases, preventing them from phosphorylating specific proteins and disrupting intracellular signaling pathways. This targeted approach inhibits the uncontrolled growth and proliferation of cancer cells, ultimately leading to their death.

The development of protein kinase inhibitors has revolutionized cancer treatment by providing more effective and less toxic alternatives to traditional chemotherapy. These drugs have demonstrated impressive results in the treatment of various cancers, including lung, breast, and leukemia.

The pharmaceutical industry invests heavily in research and development to discover novel protein kinase inhibitors with improved potency, selectivity, and pharmacokinetic properties. High-throughput screening, computational modeling, and structure-activity relationship studies are employed to identify potential lead compounds.

The success of protein kinase inhibitors in treating cancer has spurred significant interest in this subcategory of APIs. Ongoing research aims to expand their applications to other diseases, such as autoimmune disorders and neurological conditions.

In conclusion, protein kinase inhibitors are a valuable class of pharmaceutical APIs with immense potential for targeted cancer therapies. Continued advancements in this field hold promise for improved treatment outcomes and enhanced patient care.

NameCAS numberCategoryAmount of suppliersAPI market price
Abemaciclib1231929-97-7Protein kinase inhibitorsView 8 Suppliers Average price per kg: $
Abrocitnib1802446-37-1Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Adagrasib1703748-89-3Protein kinase inhibitorsView 3 Suppliers Average price per kg: $
Afatinib850140-72-6Protein kinase inhibitorsView 9 Suppliers Average price per kg: $
AlectinibProtein kinase inhibitorsView 6 Suppliers Average price per kg: $
Asciminib149632-96-9Protein kinase inhibitorsView 3 Suppliers Average price per kg: $
Axitinib319460-85-0Protein kinase inhibitorsView 13 Suppliers Average price per kg: $
Binimetinib606143-89-9Protein kinase inhibitorsView 1 Suppliers Average price per kg: $
Bosutinib380843-75-4Protein kinase inhibitorsView 7 Suppliers Average price per kg: $
Cabozantinib849217-68-1Protein kinase inhibitorsView 9 Suppliers Average price per kg: $
Cobimetinib934660-93-2Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
DabrafenibProtein kinase inhibitorsView 3 Suppliers Average price per kg: $
Encorafenib1269440-17-6Protein kinase inhibitorsView 1 Suppliers Average price per kg: $
Erlotinib183321-74-6Protein kinase inhibitorsView 39 Suppliers Average price per kg: $
Gefitinib184475-35-2Protein kinase inhibitorsView 25 Suppliers Average price per kg: $
Ibrutinib936563-96-1Protein kinase inhibitorsView 24 Suppliers Average price per kg: $
Icotinib hydrochloride186497-07-4Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Idelalisib870281-82-6Protein kinase inhibitorsView 4 Suppliers Average price per kg: $
Imatinib Mesylate152459-95-5Protein kinase inhibitorsView 47 Suppliers Average price per kg: $
Lapatinib231277-92-2Protein kinase inhibitorsView 11 Suppliers Average price per kg: $
Lenvatinib417716-92-8Protein kinase inhibitorsView 15 Suppliers Average price per kg: $
Lerociclib1628256-23-4Protein kinase inhibitorsView 1 Suppliers Average price per kg: $
Midostaurin120685-11-2Protein kinase inhibitorsView 5 Suppliers Average price per kg: $
Nilotinib641571-10-0Protein kinase inhibitorsView 17 Suppliers Average price per kg: $
Nilotinib hydrochloride anhydrous923288-95-3Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Nintedanib656247-17-5Protein kinase inhibitorsView 16 Suppliers Average price per kg: $
Olaparib763113-22-0Protein kinase inhibitorsView 13 Suppliers Average price per kg: $
Osimertinib1421373-65-0Protein kinase inhibitorsView 12 Suppliers Average price per kg: $
Palbociclib571190-30-2Protein kinase inhibitorsView 33 Suppliers Average price per kg: $
Panobinostat404950-80-7Protein kinase inhibitorsView 4 Suppliers Average price per kg: $
Pazopanib444731-52-6Protein kinase inhibitorsView 15 Suppliers Average price per kg: $
Ponatinib943319-70-8Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Regorafenib755037-03-7Protein kinase inhibitorsView 6 Suppliers Average price per kg: $
Ribociclib1211441-98-3Protein kinase inhibitorsView 7 Suppliers Average price per kg: $
Ripretinib170729-80-3Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Ruxolitinib941678-49-5Protein kinase inhibitorsView 9 Suppliers Average price per kg: $
Sonidegib956697-53-3Protein kinase inhibitorsView 3 Suppliers Average price per kg: $
Sorafenib284461-73-0Protein kinase inhibitorsView 23 Suppliers Average price per kg: $
Sotorasib1610526-40-8Protein kinase inhibitorsView 3 Suppliers Average price per kg: $
Sunitinib557795-19-4Protein kinase inhibitorsView 19 Suppliers Average price per kg: $
Tepotinib1353550-13-6Protein kinase inhibitorsView 1 Suppliers Average price per kg: $
Trametinib871700-17-3Protein kinase inhibitorsView 5 Suppliers Average price per kg: $
Tucatinib937263-43-9Protein kinase inhibitorsView 2 Suppliers Average price per kg: $
Valemetostat1809336-39-7Protein kinase inhibitorsView 1 Suppliers Average price per kg: $
Veliparib912444-00-9Protein kinase inhibitorsView 2 Suppliers Average price per kg: $