Epicriptine API Manufacturers

General Description:

Epicriptine, identified by CAS number 88660-47-3, is a notable compound with significant therapeutic applications. Epicriptine is also known as beta-dihydroergocryptine presents a molecular formula of 9,10 alpha-dihydro-13'-epi-b-ergocryptine. Together with the alpha-dihydroergocryptine, it represents one-third of the ergoloid mesylate mixture. Epicriptine differs from the alpha form on the position of one methyl group. To know more about the mixture please visit

Indications:

This drug is primarily indicated for: Please refer to and to know more about the isomer please refer to . Its use in specific medical scenarios underscores its importance in the therapeutic landscape.

Metabolism:

Epicriptine undergoes metabolic processing primarily in: Please refer to and to know more about the isomer please refer to . This metabolic pathway ensures efficient processing of the drug, helping to minimize potential toxicity and side effects.

Absorption:

The absorption characteristics of Epicriptine are crucial for its therapeutic efficacy: Please refer to and to know more about the isomer please refer to . The drug's ability to rapidly penetrate into cells ensures quick onset of action.

Half-life:

The half-life of Epicriptine is an important consideration for its dosing schedule: Please refer to and to know more about the isomer please refer to . This determines the duration of action and helps in formulating effective dosing regimens.

Protein Binding:

Epicriptine exhibits a strong affinity for binding with plasma proteins: Please refer to and to know more about the isomer please refer to . This property plays a key role in the drug's pharmacokinetics and distribution within the body.

Route of Elimination:

The elimination of Epicriptine from the body primarily occurs through: Please refer to and to know more about the isomer please refer to . Understanding this pathway is essential for assessing potential drug accumulation and toxicity risks.

Volume of Distribution:

Epicriptine is distributed throughout the body with a volume of distribution of: Please refer to and to know more about the isomer please refer to . This metric indicates how extensively the drug permeates into body tissues.

Clearance:

The clearance rate of Epicriptine is a critical factor in determining its safe and effective dosage: Please refer to and to know more about the isomer please refer to . It reflects the efficiency with which the drug is removed from the systemic circulation.

Pharmacodynamics:

Epicriptine exerts its therapeutic effects through: Please refer to and to know more about the isomer please refer to . The drug's ability to modulate various physiological processes underscores its efficacy in treating specific conditions.

Mechanism of Action:

Epicriptine functions by: Epicriptine effect is mainly due to the agonistic activity on dopamine receptor. This activity is categorized as part of the ergoline class which is defined as a producer of a vasoconstrictive effect. Please refer to and to know more about the isomer please refer to . This mechanism highlights the drug's role in inhibiting or promoting specific biological pathways, contributing to its therapeutic effects.

Toxicity:

Categories:

Epicriptine is categorized under the following therapeutic classes: Alkaloids, Dopamine Agonists. These classifications highlight the drug's diverse therapeutic applications and its importance in treating various conditions.

Experimental Properties:

Further physical and chemical characteristics of Epicriptine include:

• Boiling Point: 848 ºC at 760 mm Hg