Antineoplastics


Antineoplastics are a crucial category of pharmaceutical active pharmaceutical ingredients (APIs) primarily used in the treatment of cancer. These powerful substances inhibit or destroy the growth of cancer cells, thus impeding the progression of malignancies.

Antineoplastics exert their therapeutic effects through various mechanisms. Some APIs interfere with DNA replication, inhibiting the division and proliferation of cancer cells. Others target specific proteins or enzymes involved in tumor growth, effectively blocking their function. Additionally, certain antineoplastic agents induce programmed cell death, known as apoptosis, in cancer cells.

These APIs find application in a wide range of cancer treatments, including chemotherapy, targeted therapy, immunotherapy, and hormone therapy. They are often administered in combination with other drugs to optimize therapeutic outcomes and minimize drug resistance.

Antineoplastics are typically synthesized through complex chemical processes, ensuring high purity and potency. Stringent quality control measures are implemented throughout manufacturing to meet regulatory standards and ensure patient safety.

Although antineoplastics offer significant benefits in treating cancer, they can also cause adverse effects due to their cytotoxic nature. Common side effects include bone marrow suppression, gastrointestinal disturbances, hair loss, and immune system suppression. Close monitoring and supportive care are essential to manage these side effects effectively.

In conclusion, antineoplastics are a vital category of pharmaceutical APIs used in the treatment of cancer. Through their diverse mechanisms of action, these compounds play a critical role in combating malignancies and improving patient outcomes.

NameCAS number
10-Hydroxycamptothecin19685-09-7
2-Chloro-4-Amino-6,7-Dimethoxy quinazoline23680-84-4
2-Methoxyestradiol362-07-2
5-(1H-Pyrrol-1-yl)-1,3-dihydro-2H-benzimidazole-2-thione172152-53-3
Ansamitocin P-366584-72-3
Apaziquone114560-48-4
Aroplatin114488-24-3
Asparaginase9015-68-3
Azacitidine320-67-2
Belinostat
Bexarotene153559-49-0
Biochanin A491-80-5
Bortezomib179324-69-7
Bortezomib D-mannitol444576-08-3
Brequinar96187-53-0
Brigatinib1197953-54-0
Bropirimine56741-95-8
Bryostatin 183314-01-6
Carboplatin41575-94-4
Carfilzomib868540-17-4
Carmustine154-93-8
Ceritinib1032900-25-6
Chiauranib1256349-48-0
Cinnamaldehyde14371-10-9
Citarinostat1316215-12-9
Cladribine4291-63-8
Clofarabine123318-82-1
Combretastatin82855-09-2
Combretastatin A4117048-59-6
Coumermycin A14434-05-3
Crenolanib670220-88-9
Crizotinib877399-52-5
Dactinomycin50-76-0
Dactolisib915019-65-7
Daidzein486-66-8
Dexrazoxane24584-09-6
Dianhydrogalactitol23261-20-3
Diaziquone57998-68-2
Didox69839-83-4
Dihematoporphyrin ether97067-70-4
Docetaxel114977-28-5
Dordaviprone1616632-77-9
Droloxifene82413-20-5
Ellipticine519-23-3
Entrectinib1108743-60-7
Epichlorohydrin106-89-8
Epigallocatechin gallate989-51-5
Epofolate958646-17-8
Epothilone D189453-10-9
Eribulin253128-41-5
Esrtamustine Sodium Phosphate
Estramustine2998-57-4
Estramustine phosphate4891-15-0
Etanidazole22668-01-5
Exemestane107868-30-4
Fadrozole102676-47-1
Filanesib885060-09-3
Fimepinostat1339928-25-4
Fludarabine21679-14-1
Fluorouracil51-21-8
Fosbretabulin222030-63-9
Ginsenoside C11021-13-9
Guadecitabine929901-49-5
Homoharringtonine26833-87-4
Ilorasertib1227939-82-3
Indisulam165668-41-7
Indole120-72-9
Indole-3-carbinol700-06-1
Iniparib160003-66-7
Irinotecan97682-44-5
Irofulven158440-71-2
Ixabepilone219989-84-1
Ixazomib1072833-77-2
Lexacalcitol131875-08-6
Liarozole115575-11-6
Lurbinectedin497871-47-3
Mafosfamide88859-04-5
Maxacalcitol103909-75-7
Merestinib1206799-15-6
Methyl 2,5-dihydroxycinnamate63177-57-1
Metoprine7761-45-7
Minnelide1254702-87-8
Minnelide free acid1254885-39-6
Mitolactol10318-26-0
Mitoxantrone65271-80-9
Monomethyl Auristatin F745017-94-1
Nadofaragene firadenovec1823059-12-6
Nanatinostat1256448-47-1
Navtemadlin1352066-68-2
Nazartinib1508250-71-2
Nedaplatin95734-82-0
Olutasidenib1887014-12-1
Onapristone96346-61-1
Ortataxel186348-23-2
Patupilone152044-54-7
Pelitinib257933-82-7
Penclomedine108030-77-9
Pentostatin53910-25-1
Perillyl alcohol18457-55-1
Phenethyl Isothiocyanate2257-09-2
Pinometostat1380288-87-8
Piritrexim72732-56-0
Platinum7440-06-4
Procarbazine671-16-9
Pyrazoloacridine99009-20-8
Rabusertib911222-45-2
Rebastinib1020172-07-9
Ribonuclease
Ricolinostat1316214-52-4
Rindopepimut1108208-65-6
Romidepsin128517-07-7
Ropidoxuridine93265-81-7
Rubitecan91421-42-0
Sagopilone305841-29-6
Salirasib162520-00-5
Salvianolic acid A96574-01-5
Sapacitabine151823-14-2
Saracatinib379231-04-6
Scriptaid287383-59-9
Semaxanib194413-58-6
Seviteronel1610537-15-9
Sizofiran9050-67-3
Sodium butyrate156-54-7
Sodium phosphate P 327635-46-3
Sulforaphane142825-10-3
Talaporfin110230-98-3
Taselisib1282512-48-4
Tegafur17902-23-7
Temsirolimus162635-04-3
Teniposide29767-20-2
Tesevatinib781613-23-8
Tezacitabine171176-43-5
Tipiracil183204-74-2
Tocladesine41941-56-4
Trabedersen925681-61-4
Transcrocetinate27876-94-4
Tretamine51-18-3
Umbralisib1532533-67-7
Uracil66-22-8
Vadimezan117570-53-3
Valrubicin56124-62-0
Voruciclib1000023-04-0
Xanthohumol6754-58-1
Zelavespib873436-91-0