Antineoplastics


Antineoplastics are a crucial category of pharmaceutical active pharmaceutical ingredients (APIs) primarily used in the treatment of cancer. These powerful substances inhibit or destroy the growth of cancer cells, thus impeding the progression of malignancies.

Antineoplastics exert their therapeutic effects through various mechanisms. Some APIs interfere with DNA replication, inhibiting the division and proliferation of cancer cells. Others target specific proteins or enzymes involved in tumor growth, effectively blocking their function. Additionally, certain antineoplastic agents induce programmed cell death, known as apoptosis, in cancer cells.

These APIs find application in a wide range of cancer treatments, including chemotherapy, targeted therapy, immunotherapy, and hormone therapy. They are often administered in combination with other drugs to optimize therapeutic outcomes and minimize drug resistance.

Antineoplastics are typically synthesized through complex chemical processes, ensuring high purity and potency. Stringent quality control measures are implemented throughout manufacturing to meet regulatory standards and ensure patient safety.

Although antineoplastics offer significant benefits in treating cancer, they can also cause adverse effects due to their cytotoxic nature. Common side effects include bone marrow suppression, gastrointestinal disturbances, hair loss, and immune system suppression. Close monitoring and supportive care are essential to manage these side effects effectively.

In conclusion, antineoplastics are a vital category of pharmaceutical APIs used in the treatment of cancer. Through their diverse mechanisms of action, these compounds play a critical role in combating malignancies and improving patient outcomes.

NameCAS numberCategoryAmount of suppliersAPI market price
10-Hydroxycamptothecin19685-09-7AntineoplasticsView 2 Suppliers Average price per kg: $
2-Chloro-4-Amino-6,7-Dimethoxy quinazoline23680-84-4AntineoplasticsView 1 Suppliers Average price per kg: $
2-Methoxyestradiol362-07-2AntineoplasticsView 1 Suppliers Average price per kg: $
5-(1H-Pyrrol-1-yl)-1,3-dihydro-2H-benzimidazole-2-thione172152-53-3AntineoplasticsView 1 Suppliers Average price per kg: $
Ansamitocin P-366584-72-3AntineoplasticsView 1 Suppliers Average price per kg: $
Apaziquone114560-48-4AntineoplasticsView 0 Suppliers Average price per kg: $
Aroplatin114488-24-3AntineoplasticsView 0 Suppliers Average price per kg: $
Asparaginase9015-68-3AntineoplasticsView 4 Suppliers Average price per kg: $
Azacitidine320-67-2AntineoplasticsView 28 Suppliers Average price per kg: $
BelinostatAntineoplasticsView 5 Suppliers Average price per kg: $
Bexarotene153559-49-0AntineoplasticsView 7 Suppliers Average price per kg: $
Biochanin A491-80-5AntineoplasticsView 0 Suppliers Average price per kg: $
Bortezomib179324-69-7AntineoplasticsView 41 Suppliers Average price per kg: $
Bortezomib D-mannitol444576-08-3AntineoplasticsView 0 Suppliers Average price per kg: $
Brequinar96187-53-0AntineoplasticsView 0 Suppliers Average price per kg: $
Brigatinib1197953-54-0AntineoplasticsView 0 Suppliers Average price per kg: $
Bropirimine56741-95-8AntineoplasticsView 0 Suppliers Average price per kg: $
Bryostatin 183314-01-6AntineoplasticsView 0 Suppliers Average price per kg: $
Carboplatin41575-94-4AntineoplasticsView 27 Suppliers Average price per kg: $
Carfilzomib868540-17-4AntineoplasticsView 19 Suppliers Average price per kg: $
Carmustine154-93-8AntineoplasticsView 12 Suppliers Average price per kg: $
Ceritinib1032900-25-6AntineoplasticsView 3 Suppliers Average price per kg: $
Chiauranib1256349-48-0AntineoplasticsView 0 Suppliers Average price per kg: $
Cinnamaldehyde14371-10-9AntineoplasticsView 0 Suppliers Average price per kg: $
Citarinostat1316215-12-9AntineoplasticsView 0 Suppliers Average price per kg: $
Cladribine4291-63-8AntineoplasticsView 6 Suppliers Average price per kg: $
Clofarabine123318-82-1AntineoplasticsView 15 Suppliers Average price per kg: $
Combretastatin82855-09-2AntineoplasticsView 0 Suppliers Average price per kg: $
Combretastatin A4117048-59-6AntineoplasticsView 0 Suppliers Average price per kg: $
Coumermycin A14434-05-3AntineoplasticsView 0 Suppliers Average price per kg: $
Crenolanib670220-88-9AntineoplasticsView 0 Suppliers Average price per kg: $
Crizotinib877399-52-5AntineoplasticsView 9 Suppliers Average price per kg: $
Dactinomycin50-76-0AntineoplasticsView 2 Suppliers Average price per kg: $
Dactolisib915019-65-7AntineoplasticsView 0 Suppliers Average price per kg: $
Daidzein486-66-8AntineoplasticsView 0 Suppliers Average price per kg: $
Dexrazoxane24584-09-6AntineoplasticsView 8 Suppliers Average price per kg: $
Dianhydrogalactitol23261-20-3AntineoplasticsView 0 Suppliers Average price per kg: $
Diaziquone57998-68-2AntineoplasticsView 0 Suppliers Average price per kg: $
Didox69839-83-4AntineoplasticsView 0 Suppliers Average price per kg: $
Dihematoporphyrin ether97067-70-4AntineoplasticsView 0 Suppliers Average price per kg: $
Docetaxel114977-28-5AntineoplasticsView 46 Suppliers Average price per kg: $
Dordaviprone1616632-77-9AntineoplasticsView 0 Suppliers Average price per kg: $
Droloxifene82413-20-5AntineoplasticsView 0 Suppliers Average price per kg: $
Ellipticine519-23-3AntineoplasticsView 0 Suppliers Average price per kg: $
Entrectinib1108743-60-7AntineoplasticsView 1 Suppliers Average price per kg: $
Epichlorohydrin106-89-8AntineoplasticsView 2 Suppliers Average price per kg: $
Epigallocatechin gallate989-51-5AntineoplasticsView 0 Suppliers Average price per kg: $
Epofolate958646-17-8AntineoplasticsView 0 Suppliers Average price per kg: $
Epothilone D189453-10-9AntineoplasticsView 0 Suppliers Average price per kg: $
Eribulin253128-41-5AntineoplasticsView 5 Suppliers Average price per kg: $
Esrtamustine Sodium PhosphateAntineoplasticsView 1 Suppliers Average price per kg: $
Estramustine2998-57-4AntineoplasticsView 4 Suppliers Average price per kg: $
Estramustine phosphate4891-15-0AntineoplasticsView 0 Suppliers Average price per kg: $
Etanidazole22668-01-5AntineoplasticsView 0 Suppliers Average price per kg: $
Exemestane107868-30-4AntineoplasticsView 26 Suppliers Average price per kg: $
Fadrozole102676-47-1AntineoplasticsView 0 Suppliers Average price per kg: $
Filanesib885060-09-3AntineoplasticsView 0 Suppliers Average price per kg: $
Fimepinostat1339928-25-4AntineoplasticsView 0 Suppliers Average price per kg: $
Fludarabine21679-14-1AntineoplasticsView 12 Suppliers Average price per kg: $
Fluorouracil51-21-8AntineoplasticsView 11 Suppliers Average price per kg: $
Fosbretabulin222030-63-9AntineoplasticsView 0 Suppliers Average price per kg: $
Ginsenoside C11021-13-9AntineoplasticsView 0 Suppliers Average price per kg: $
Guadecitabine929901-49-5AntineoplasticsView 0 Suppliers Average price per kg: $
Homoharringtonine26833-87-4AntineoplasticsView 1 Suppliers Average price per kg: $
Ilorasertib1227939-82-3AntineoplasticsView 0 Suppliers Average price per kg: $
Indisulam165668-41-7AntineoplasticsView 0 Suppliers Average price per kg: $
Indole120-72-9AntineoplasticsView 1 Suppliers Average price per kg: $
Indole-3-carbinol700-06-1AntineoplasticsView 0 Suppliers Average price per kg: $
Iniparib160003-66-7AntineoplasticsView 0 Suppliers Average price per kg: $
Irinotecan97682-44-5AntineoplasticsView 33 Suppliers Average price per kg: $
Irofulven158440-71-2AntineoplasticsView 0 Suppliers Average price per kg: $
Ixabepilone219989-84-1AntineoplasticsView 1 Suppliers Average price per kg: $
Ixazomib1072833-77-2AntineoplasticsView 6 Suppliers Average price per kg: $
Lexacalcitol131875-08-6AntineoplasticsView 0 Suppliers Average price per kg: $
Liarozole115575-11-6AntineoplasticsView 0 Suppliers Average price per kg: $
Lurbinectedin497871-47-3AntineoplasticsView 5 Suppliers Average price per kg: $
Mafosfamide88859-04-5AntineoplasticsView 0 Suppliers Average price per kg: $
Maxacalcitol103909-75-7AntineoplasticsView 3 Suppliers Average price per kg: $
Merestinib1206799-15-6AntineoplasticsView 0 Suppliers Average price per kg: $
Methyl 2,5-dihydroxycinnamate63177-57-1AntineoplasticsView 0 Suppliers Average price per kg: $
Metoprine7761-45-7AntineoplasticsView 0 Suppliers Average price per kg: $
Minnelide1254702-87-8AntineoplasticsView 0 Suppliers Average price per kg: $
Minnelide free acid1254885-39-6AntineoplasticsView 0 Suppliers Average price per kg: $
Mitolactol10318-26-0AntineoplasticsView 0 Suppliers Average price per kg: $
Mitoxantrone65271-80-9AntineoplasticsView 7 Suppliers Average price per kg: $
Monomethyl Auristatin F745017-94-1AntineoplasticsView 2 Suppliers Average price per kg: $
Nadofaragene firadenovec1823059-12-6AntineoplasticsView 0 Suppliers Average price per kg: $
Nanatinostat1256448-47-1AntineoplasticsView 0 Suppliers Average price per kg: $
Navtemadlin1352066-68-2AntineoplasticsView 0 Suppliers Average price per kg: $
Nazartinib1508250-71-2AntineoplasticsView 0 Suppliers Average price per kg: $
Nedaplatin95734-82-0AntineoplasticsView 1 Suppliers Average price per kg: $
Olutasidenib1887014-12-1AntineoplasticsView 0 Suppliers Average price per kg: $
Onapristone96346-61-1AntineoplasticsView 0 Suppliers Average price per kg: $
Ortataxel186348-23-2AntineoplasticsView 0 Suppliers Average price per kg: $
Patupilone152044-54-7AntineoplasticsView 0 Suppliers Average price per kg: $
Pelitinib257933-82-7AntineoplasticsView 0 Suppliers Average price per kg: $
Penclomedine108030-77-9AntineoplasticsView 0 Suppliers Average price per kg: $
Pentostatin53910-25-1AntineoplasticsView 3 Suppliers Average price per kg: $
Perillyl alcohol18457-55-1AntineoplasticsView 0 Suppliers Average price per kg: $
Phenethyl Isothiocyanate2257-09-2AntineoplasticsView 0 Suppliers Average price per kg: $
Pinometostat1380288-87-8AntineoplasticsView 0 Suppliers Average price per kg: $
Piritrexim72732-56-0AntineoplasticsView 0 Suppliers Average price per kg: $
Platinum7440-06-4AntineoplasticsView 0 Suppliers Average price per kg: $
Procarbazine671-16-9AntineoplasticsView 3 Suppliers Average price per kg: $
Pyrazoloacridine99009-20-8AntineoplasticsView 0 Suppliers Average price per kg: $
Rabusertib911222-45-2AntineoplasticsView 0 Suppliers Average price per kg: $
Rebastinib1020172-07-9AntineoplasticsView 0 Suppliers Average price per kg: $
RibonucleaseAntineoplasticsView 2 Suppliers Average price per kg: $
Ricolinostat1316214-52-4AntineoplasticsView 0 Suppliers Average price per kg: $
Rindopepimut1108208-65-6AntineoplasticsView 0 Suppliers Average price per kg: $
Romidepsin128517-07-7AntineoplasticsView 6 Suppliers Average price per kg: $
Ropidoxuridine93265-81-7AntineoplasticsView 0 Suppliers Average price per kg: $
Rubitecan91421-42-0AntineoplasticsView 0 Suppliers Average price per kg: $
Sagopilone305841-29-6AntineoplasticsView 0 Suppliers Average price per kg: $
Salirasib162520-00-5AntineoplasticsView 0 Suppliers Average price per kg: $
Salvianolic acid A96574-01-5AntineoplasticsView 0 Suppliers Average price per kg: $
Sapacitabine151823-14-2AntineoplasticsView 0 Suppliers Average price per kg: $
Saracatinib379231-04-6AntineoplasticsView 0 Suppliers Average price per kg: $
Scriptaid287383-59-9AntineoplasticsView 0 Suppliers Average price per kg: $
Semaxanib194413-58-6AntineoplasticsView 0 Suppliers Average price per kg: $
Seviteronel1610537-15-9AntineoplasticsView 0 Suppliers Average price per kg: $
Sizofiran9050-67-3AntineoplasticsView 0 Suppliers Average price per kg: $
Sodium butyrate156-54-7AntineoplasticsView 1 Suppliers Average price per kg: $
Sodium phosphate P 327635-46-3AntineoplasticsView 0 Suppliers Average price per kg: $
Sulforaphane142825-10-3AntineoplasticsView 0 Suppliers Average price per kg: $
Talaporfin110230-98-3AntineoplasticsView 0 Suppliers Average price per kg: $
Taselisib1282512-48-4AntineoplasticsView 0 Suppliers Average price per kg: $
Tegafur17902-23-7AntineoplasticsView 3 Suppliers Average price per kg: $
Temsirolimus162635-04-3AntineoplasticsView 8 Suppliers Average price per kg: $
Teniposide29767-20-2AntineoplasticsView 2 Suppliers Average price per kg: $
Tesevatinib781613-23-8AntineoplasticsView 0 Suppliers Average price per kg: $
Tezacitabine171176-43-5AntineoplasticsView 0 Suppliers Average price per kg: $
Tipiracil183204-74-2AntineoplasticsView 2 Suppliers Average price per kg: $
Tocladesine41941-56-4AntineoplasticsView 0 Suppliers Average price per kg: $
Trabedersen925681-61-4AntineoplasticsView 0 Suppliers Average price per kg: $
Transcrocetinate27876-94-4AntineoplasticsView 0 Suppliers Average price per kg: $
Tretamine51-18-3AntineoplasticsView 0 Suppliers Average price per kg: $
Umbralisib1532533-67-7AntineoplasticsView 0 Suppliers Average price per kg: $
Uracil66-22-8AntineoplasticsView 1 Suppliers Average price per kg: $
Vadimezan117570-53-3AntineoplasticsView 0 Suppliers Average price per kg: $
Valrubicin56124-62-0AntineoplasticsView 3 Suppliers Average price per kg: $
Voruciclib1000023-04-0AntineoplasticsView 0 Suppliers Average price per kg: $
Xanthohumol6754-58-1AntineoplasticsView 0 Suppliers Average price per kg: $
Zelavespib873436-91-0AntineoplasticsView 0 Suppliers Average price per kg: $