Antihypertensive agents


Antihypertensive agents are a crucial category of pharmaceutical active pharmaceutical ingredients (APIs) used to treat high blood pressure, also known as hypertension. These medications are designed to lower blood pressure and reduce the risk of associated cardiovascular complications.

Antihypertensive agents function by targeting various mechanisms involved in blood pressure regulation. Some common classes of antihypertensive agents include angiotensin-converting enzyme (ACE) inhibitors, angiotensin II receptor blockers (ARBs), beta-blockers, calcium channel blockers (CCBs), and diuretics.

ACE inhibitors work by inhibiting the enzyme responsible for converting angiotensin I to angiotensin II, a hormone that constricts blood vessels. ARBs, on the other hand, block the receptors to which angiotensin II binds, thereby preventing its vasoconstrictive effects.

Beta-blockers reduce blood pressure by blocking the effects of adrenaline and noradrenaline, which are responsible for increasing heart rate and constricting blood vessels. CCBs inhibit calcium from entering the smooth muscles of blood vessels, resulting in relaxation and vasodilation. Diuretics promote the elimination of excess fluid and sodium from the body, reducing blood volume and thereby lowering blood pressure.

Antihypertensive agents are typically prescribed based on the individual patient's condition and specific needs. They can be used alone or in combination to achieve optimal blood pressure control. It is important to note that antihypertensive agents should be taken regularly as prescribed by a healthcare professional and may require periodic monitoring to ensure their effectiveness and manage any potential side effects.

In summary, antihypertensive agents play a vital role in the management of hypertension by targeting various mechanisms involved in blood pressure regulation. These medications offer significant benefits in reducing the risk of cardiovascular complications associated with high blood pressure.

NameCAS numberCategoryAmount of suppliersAPI market price
Acebutolol37517-30-9Beta blockersView 5 Suppliers Average price per kg: $
Acebutolol HCl34381-68-5Beta blockersView 1 Suppliers Average price per kg: $
Acemetacin53164-05-9Antihypertensive agentsView 1 Suppliers Average price per kg: $
Acetic acid C-1178887-71-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
Aganepag isopropyl910562-20-8Antihypertensive agentsView 0 Suppliers Average price per kg: $
Alfuzosin81403-80-7Alpha blockersView 15 Suppliers Average price per kg: $
Aliskiren173334-57-1Renin inhibitorsView 4 Suppliers Average price per kg: $
Alpha Cyclohexyl Mandelic Acid Methyl Ester10399-13-0DiureticsView 1 Suppliers Average price per kg: $
Alprostadil745-65-3VasodilatorsView 14 Suppliers Average price per kg: $
Ambrisentan177036-94-1Other antihypertensive agentsView 11 Suppliers Average price per kg: $
Amiloride2609-46-3DiureticsView 7 Suppliers Average price per kg: $
Amitraz33089-61-1Antihypertensive agentsView 1 Suppliers Average price per kg: $
Amitriptylinoxide4317-14-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Amlodipine88150-42-9Calcium Channel BlockersView 71 Suppliers Average price per kg: $
Amlodipine BesilateCalcium Channel BlockersView 10 Suppliers Average price per kg: $
Apraclonidine66711-21-5Alpha-2 adrenergic agonistView 3 Suppliers Average price per kg: $
Aprocitentan1103522-45-7Antihypertensive agentsView 1 Suppliers Average price per kg: $
Arotinolol68377-92-4Beta blockersView 1 Suppliers Average price per kg: $
Atenolol29122-68-7Beta blockersView 26 Suppliers Average price per kg: $
Atipamezole104075-48-1Alpha blockersView 3 Suppliers Average price per kg: $
Avanafil330784-47-9DiureticsView 9 Suppliers Average price per kg: $
Azapetine146-36-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Azelnidipine123524-52-7Calcium Channel BlockersView 7 Suppliers Average price per kg: $
Azilsartan medoxomil863031-21-4Angiotensin Receptor BlockersView 19 Suppliers Average price per kg: $
Azosemide27589-33-9DiureticsView 4 Suppliers Average price per kg: $
Barnidipine104713-75-9Calcium Channel BlockersView 2 Suppliers Average price per kg: $
Benazepril86541-75-5ACE inhibitorsView 17 Suppliers Average price per kg: $
Bendroflumethiazide73-48-3DiureticsView 5 Suppliers Average price per kg: $
Benidipine105979-17-7Calcium Channel BlockersView 8 Suppliers Average price per kg: $
Benzthiazide91-33-8DiureticsView 1 Suppliers Average price per kg: $
Benzyl Nicotinate94-44-0VasodilatorsView 4 Suppliers Average price per kg: $
Betaxolol63659-18-7Beta blockersView 12 Suppliers Average price per kg: $
Bevantolol59170-23-9Beta blockersView 1 Suppliers Average price per kg: $
Bietaserpine53-18-9Antihypertensive agentsView 0 Suppliers Average price per kg: $
Bisoprolol66722-44-9Beta blockersView 37 Suppliers Average price per kg: $
Bosentan147536-97-8VasodilatorsView 42 Suppliers Average price per kg: $
Buflomedil55837-25-7Antihypertensive agentsView 0 Suppliers Average price per kg: $
Bumetanide28395-03-1DiureticsView 10 Suppliers Average price per kg: $
Buthiazide2043-38-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Cadralazine64241-34-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
Candesartan139481-59-7Angiotensin Receptor BlockersView 53 Suppliers Average price per kg: $
Canrenone976-71-6Antihypertensive agentsView 0 Suppliers Average price per kg: $
Captopril62571-86-2ACE inhibitorsView 23 Suppliers Average price per kg: $
Carrot seedDiureticsView 1 Suppliers Average price per kg: $
Carteolol51781-06-7Beta blockersView 5 Suppliers Average price per kg: $
Carvedilol72956-09-3Beta blockersView 49 Suppliers Average price per kg: $
Carvedilol phosphate hemihydrate851220-85-4Alpha blockersView 2 Suppliers Average price per kg: $
Celery seedDiureticsView 1 Suppliers Average price per kg: $
Celiprolol56980-93-9Beta blockersView 4 Suppliers Average price per kg: $
Chlorothiazide58-94-6DiureticsView 4 Suppliers Average price per kg: $
Chlorthalidone77-36-1DiureticsView 19 Suppliers Average price per kg: $
Cicletanine89943-82-8Antihypertensive agentsView 0 Suppliers Average price per kg: $
Cilazapril88768-40-5ACE inhibitorsView 6 Suppliers Average price per kg: $
Cilnidipine132203-70-4Calcium Channel BlockersView 11 Suppliers Average price per kg: $
Clevidipine167221-71-8Calcium Channel BlockersView 2 Suppliers Average price per kg: $
Clofenamide671-95-4Antihypertensive agentsView 0 Suppliers Average price per kg: $
Clonidine4205-90-7Antihypertensive agentsView 13 Suppliers Average price per kg: $
Clopamide636-54-4DiureticsView 1 Suppliers Average price per kg: $
Cloranolol39563-28-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
Clorgiline17780-72-2Antihypertensive agentsView 0 Suppliers Average price per kg: $
Cloridarol3611-72-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Cyclopenthiazide742-20-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Cyclopentyl Mandelic Acid427-49-6DiureticsView 1 Suppliers Average price per kg: $
Dapiprazole72822-12-9Alpha blockersView 1 Suppliers Average price per kg: $
Deoxyepinephrine501-15-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
DetomidineAlpha-2 adrenergic agonistView 3 Suppliers Average price per kg: $
Dexmedetomidine113775-47-6Alpha-2 adrenergic agonistView 19 Suppliers Average price per kg: $
Dexniguldipine120054-86-6Antihypertensive agentsView 0 Suppliers Average price per kg: $
Diclofenamide120-97-8DiureticsView 4 Suppliers Average price per kg: $
Diethylnorspermine121749-39-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Dihydralazine484-23-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Diltiazem42399-41-7Calcium Channel BlockersView 20 Suppliers Average price per kg: $
Doxazosin74191-85-8Alpha blockersView 25 Suppliers Average price per kg: $
Efonidipine111011-63-3Calcium Channel BlockersView 2 Suppliers Average price per kg: $
Enalapril75847-73-3ACE inhibitorsView 19 Suppliers Average price per kg: $
EnalaprilatACE inhibitorsView 2 Suppliers Average price per kg: $
Endralazine39715-02-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Epanolol86880-51-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
Epitizide1764-85-8Antihypertensive agentsView 0 Suppliers Average price per kg: $
Eplerenone107724-20-9Aldosterone antagonistsView 12 Suppliers Average price per kg: $
Epoprostenol35121-78-9VasodilatorsView 10 Suppliers Average price per kg: $
Eprosartan133040-01-4Angiotensin Receptor BlockersView 8 Suppliers Average price per kg: $
Esatenolol93379-54-5Antihypertensive agentsView 0 Suppliers Average price per kg: $
Esaxerenone1632006-28-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Esmolol81147-92-4Beta blockersView 10 Suppliers Average price per kg: $
Etacrynic acid58-54-8DiureticsView 14 Suppliers Average price per kg: $
Ethyl 4-(2-Hydroxy-2-Propyl)-2-Propyl-1H-Imidazole-5-Carboxylate144689-93-0Antihypertensive agentsView 1 Suppliers Average price per kg: $
Felodipine72509-76-3Calcium Channel BlockersView 13 Suppliers Average price per kg: $
Fenoldopam67227-56-9Antihypertensive agentsView 3 Suppliers Average price per kg: $
Fenozolone15302-16-6Antihypertensive agentsView 0 Suppliers Average price per kg: $
Finerenone1050477-31-0Aldosterone antagonistsView 8 Suppliers Average price per kg: $
Flunarizine52468-60-7Calcium Channel BlockersView 13 Suppliers Average price per kg: $
Fosinopril98048-97-6ACE inhibitorsView 7 Suppliers Average price per kg: $
Furosemide54-31-9DiureticsView 30 Suppliers Average price per kg: $
Gepefrine18840-47-6Antihypertensive agentsView 0 Suppliers Average price per kg: $
Guanazodine32059-15-7Antihypertensive agentsView 0 Suppliers Average price per kg: $
Guanfacine29110-47-2Alpha-2 adrenergic agonistView 6 Suppliers Average price per kg: $
Guanoclor5001-32-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Guanoxabenz24047-25-4Antihypertensive agentsView 0 Suppliers Average price per kg: $
Guanoxan2165-19-7Antihypertensive agentsView 0 Suppliers Average price per kg: $
Heather flowerDiureticsView 1 Suppliers Average price per kg: $
Heather herbDiureticsView 1 Suppliers Average price per kg: $
Heptaminol hydrochloride543-15-7VasodilatorsView 1 Suppliers Average price per kg: $
HistamineVasodilatorsView 2 Suppliers Average price per kg: $
Histamine Phosphate51-74-1VasodilatorsView 5 Suppliers Average price per kg: $
Histamine dihydrochloride56-92-8VasodilatorsView 8 Suppliers Average price per kg: $
Hydralazine86-54-4VasodilatorsView 13 Suppliers Average price per kg: $
Hydrochlorothiazide58-93-5DiureticsView 35 Suppliers Average price per kg: $
Hydroflumethiazide135-09-1DiureticsView 1 Suppliers Average price per kg: $
Idazoxan79944-58-4Antihypertensive agentsView 0 Suppliers Average price per kg: $
Indapamide26807-65-8DiureticsView 22 Suppliers Average price per kg: $
Indobufen63610-08-2Antihypertensive agentsView 0 Suppliers Average price per kg: $
Indoramin26844-12-2Alpha blockersView 1 Suppliers Average price per kg: $
Iofetamine I-12375917-92-9Antihypertensive agentsView 0 Suppliers Average price per kg: $
Irbesartan138402-11-6Angiotensin Receptor BlockersView 60 Suppliers Average price per kg: $
Isradipine75695-93-1Calcium Channel BlockersView 7 Suppliers Average price per kg: $
Ketanserin74050-98-9Antihypertensive agentsView 1 Suppliers Average price per kg: $
Labetalol36894-69-6Beta blockersView 14 Suppliers Average price per kg: $
Lacidipine103890-78-4Calcium Channel BlockersView 11 Suppliers Average price per kg: $
Lercanidipine100427-26-7Calcium Channel BlockersView 12 Suppliers Average price per kg: $
Levamlodipine103129-82-4Calcium Channel BlockersView 1 Suppliers Average price per kg: $
Levobunolol47141-42-4Beta blockersView 4 Suppliers Average price per kg: $
Linsidomine33876-97-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Lisinopril83915-83-7ACE inhibitorsView 17 Suppliers Average price per kg: $
Lofexidine31036-80-3Alpha blockersView 1 Suppliers Average price per kg: $
Lonazolac53808-88-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Losartan Potassium114798-26-4Angiotensin Receptor BlockersView 60 Suppliers Average price per kg: $
Macitentan441798-33-0Other antihypertensive agentsView 15 Suppliers Average price per kg: $
Manidipine89226-50-6Calcium Channel BlockersView 4 Suppliers Average price per kg: $
Mannitol69-65-8DiureticsView 17 Suppliers Average price per kg: $
Mebutizide3568-00-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Medetomidine86347-14-0Alpha-2 adrenergic agonistView 3 Suppliers Average price per kg: $
Mefenorex17243-57-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Mefruside7195-27-9Antihypertensive agentsView 0 Suppliers Average price per kg: $
Mephedrone1189805-46-6Antihypertensive agentsView 0 Suppliers Average price per kg: $
Mepindolol23694-81-7Antihypertensive agentsView 0 Suppliers Average price per kg: $
Metergoline17692-51-2Antihypertensive agentsView 0 Suppliers Average price per kg: $
Methoserpidine865-04-3Antihypertensive agentsView 0 Suppliers Average price per kg: $
Methyclothiazide135-07-9DiureticsView 1 Suppliers Average price per kg: $
Methyl Nicotinate93-60-7VasodilatorsView 6 Suppliers Average price per kg: $
Methyldopa555-30-6Antihypertensive agentsView 12 Suppliers Average price per kg: $
Metolazone17560-51-9DiureticsView 5 Suppliers Average price per kg: $
Metoprolol51384-51-1Beta blockersView 40 Suppliers Average price per kg: $
Minoxidil38304-91-5VasodilatorsView 37 Suppliers Average price per kg: $
Moexipril103775-10-6ACE inhibitorsView 3 Suppliers Average price per kg: $
Molsidomine25717-80-0VasodilatorsView 2 Suppliers Average price per kg: $
Moxonidine75438-57-2Antihypertensive agentsView 11 Suppliers Average price per kg: $
Muzolimine55294-15-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Nadolol42200-33-9Beta blockersView 8 Suppliers Average price per kg: $
Naftopidil57149-07-2Antihypertensive agentsView 1 Suppliers Average price per kg: $
Naphazoline835-31-4Alpha blockersView 9 Suppliers Average price per kg: $
Nebivolol118457-14-0Beta blockersView 22 Suppliers Average price per kg: $
Nicardipine55985-32-5Calcium Channel BlockersView 13 Suppliers Average price per kg: $
Nifedipine21829-25-4Calcium Channel BlockersView 28 Suppliers Average price per kg: $
Nilvadipine75530-68-6Calcium Channel BlockersView 4 Suppliers Average price per kg: $
Nimodipine66085-59-4Calcium Channel BlockersView 17 Suppliers Average price per kg: $
Nisoldipine63675-72-9Calcium Channel BlockersView 8 Suppliers Average price per kg: $
Nitrendipine39562-70-4Calcium Channel BlockersView 5 Suppliers Average price per kg: $
Nitric Oxide10102-43-9VasodilatorsView 3 Suppliers Average price per kg: $
Nitroglycerin55-63-0VasodilatorsView 3 Suppliers Average price per kg: $
Nitroprusside15078-28-1VasodilatorsView 3 Suppliers Average price per kg: $
Olmesartan144689-24-7Angiotensin Receptor BlockersView 76 Suppliers Average price per kg: $
Pamabrom606-04-2DiureticsView 5 Suppliers Average price per kg: $
Papaverine58-74-2VasodilatorsView 11 Suppliers Average price per kg: $
Penbutolol38363-40-5Beta blockersView 1 Suppliers Average price per kg: $
Perindopril82834-16-0ACE inhibitorsView 25 Suppliers Average price per kg: $
Phenoxybenzamine59-96-1Alpha blockersView 6 Suppliers Average price per kg: $
Phentolamine50-60-2Alpha blockersView 8 Suppliers Average price per kg: $
Pinacidil60560-33-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Pindolol13523-86-9Beta blockersView 3 Suppliers Average price per kg: $
Piretanide55837-27-9DiureticsView 2 Suppliers Average price per kg: $
Prazosin19216-56-9Alpha blockersView 7 Suppliers Average price per kg: $
Propranolol525-66-6Beta blockersView 19 Suppliers Average price per kg: $
Quinapril85441-61-8ACE inhibitorsView 9 Suppliers Average price per kg: $
Quinoline Yellow WS8004-92-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Ralinepag1187856-49-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Ramipril87333-19-5ACE inhibitorsView 28 Suppliers Average price per kg: $
Regadenoson313348-27-5VasodilatorsView 13 Suppliers Average price per kg: $
Reserpine50-55-5Antihypertensive agentsView 6 Suppliers Average price per kg: $
Riociguat625115-55-1sGC stimulatorView 7 Suppliers Average price per kg: $
Rostafuroxin156722-18-8Antihypertensive agentsView 0 Suppliers Average price per kg: $
Sacubitril149709-62-6ACE inhibitorsView 12 Suppliers Average price per kg: $
Salbutamol18559-94-9Beta blockersView 39 Suppliers Average price per kg: $
Salmeterol89365-50-4Beta blockersView 31 Suppliers Average price per kg: $
Saralasin34273-10-4Antihypertensive agentsView 0 Suppliers Average price per kg: $
Selexipag475086-01-2Other antihypertensive agentsView 8 Suppliers Average price per kg: $
Sepetaprost1262873-06-2Antihypertensive agentsView 0 Suppliers Average price per kg: $
Serdexmethylphenidate1996626-29-9Antihypertensive agentsView 0 Suppliers Average price per kg: $
Silodosin160970-54-7Alpha blockersView 31 Suppliers Average price per kg: $
Sotalol3930-20-9Beta blockersView 8 Suppliers Average price per kg: $
Spironolactone52-01-7DiureticsView 26 Suppliers Average price per kg: $
Talinolol57460-41-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Tamsulosin106133-20-4Alpha blockersView 51 Suppliers Average price per kg: $
Taprenepag752187-80-7Antihypertensive agentsView 0 Suppliers Average price per kg: $
Telmisartan144701-48-4Angiotensin Receptor BlockersView 84 Suppliers Average price per kg: $
Temocapril111902-57-9ACE inhibitorsView 2 Suppliers Average price per kg: $
Tenidap120210-48-2Antihypertensive agentsView 0 Suppliers Average price per kg: $
Terazosin63590-64-7Alpha blockersView 18 Suppliers Average price per kg: $
Terbogrel149979-74-8Antihypertensive agentsView 0 Suppliers Average price per kg: $
Terguride37686-84-3Antihypertensive agentsView 0 Suppliers Average price per kg: $
Tertatolol83688-84-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Tetrahydrocannabivarin31262-37-0Antihypertensive agentsView 0 Suppliers Average price per kg: $
Theodrenaline13460-98-5Antihypertensive agentsView 1 Suppliers Average price per kg: $
Timolol26839-75-8Beta blockersView 33 Suppliers Average price per kg: $
Tolonidine4201-22-3Antihypertensive agentsView 0 Suppliers Average price per kg: $
Torasemide56211-40-6DiureticsView 24 Suppliers Average price per kg: $
Trabodenoson871108-05-3Antihypertensive agentsView 0 Suppliers Average price per kg: $
Tramazoline1082-57-1Antihypertensive agentsView 0 Suppliers Average price per kg: $
Trandolapril87679-37-6ACE inhibitorsView 7 Suppliers Average price per kg: $
Treprostinil81846-19-7VasodilatorsView 13 Suppliers Average price per kg: $
Triamterene396-01-0DiureticsView 4 Suppliers Average price per kg: $
Trichlormethiazide133-67-5DiureticsView 4 Suppliers Average price per kg: $
Ubenimex58970-76-6ACE inhibitorsView 4 Suppliers Average price per kg: $
Urapidil64887-14-5Alpha blockersView 6 Suppliers Average price per kg: $
Valsartan137862-53-4Angiotensin Receptor BlockersView 53 Suppliers Average price per kg: $
Verapamil52-53-9Calcium Channel BlockersView 15 Suppliers Average price per kg: $
Vericiguat1350653-20-1sGC stimulatorView 4 Suppliers Average price per kg: $
Xanthinol2530-97-4VasodilatorsView 1 Suppliers Average price per kg: $
Xipamide14293-44-8Antihypertensive agentsView 1 Suppliers Average price per kg: $
Yohimbine146-48-5Alpha blockersView 6 Suppliers Average price per kg: $
Zamicastat1080028-80-3Antihypertensive agentsView 0 Suppliers Average price per kg: $